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CD69

Brief Information

Name:DNA (cytosine-5)-methyltransferase 1
Target Synonym:Dnmt1,AIM,MCMT,DNA methyltransferase HsaI,DNA Methyltransferase 1,CXXC-Type Zinc Finger Protein 9,DNA MTase HsaI,M.HsaI,CXXC9,EC:2.1.1.37,DNA (Cytosine-5-)-Methyltransferase 1,DNMT,DNA (Cytosine-5)-Methyltransferase 1,EC 2.1.1.37,ADCADN,HSN1E
Number of Launched Drugs:5
Number of Drugs in Clinical Trials:9
Lastest Research Phase:Approved

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Part of Bioactivity data

FABm022-01-Cell-based assay
 CD69 FACS

Flow cytometric analysis of Jurkat staining with PE-Labeled Monoclonal Anti-Human CD69 Antibody, Mouse IgG1 (3C5B7) (Cat. No. FABm022-01) at 1:20 dilution (5 μL of the antibody stock solution corresponds to labeling of 1e6 cells in a final volume of 100 µL), compared with isotype control antibody. PE signal was used to evaluate the binding activity (QC tested).

Synonym Name

CD69,CLEC2C,AIM,BL-AC/P26,EA1,GP32/28,MLR-3

Background

Early activation antigen CD69 is also known as C-type lectin domain family 2 member C (CLEC2C), Activation inducer molecule (AIM), Early T-cell activation antigen p60, Leukocyte surface antigen Leu-23. CD69 contains one C-type lectin domain. CD69 / CLEC2C is expressed on the surface of activated T-cells, B-cells, natural killer cells, neutrophils, eosinophils, epidermal Langerhans cells and platelets. CD69 is induced by antigens, mitogens or activators of PKC on the surface of T and B-lymphocytes and by interaction of IL-2 with the p75 IL-2R on the surface of NK cells. CD69 / CLEC2C involved in lymphocyte proliferation and functions as a signal transmitting receptor in lymphocytes, natural killer (NK) cells, and platelets.

Clinical and Translational Updates

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Decitabine/Cedazuridine ASTX-727-LD; ASTX-727-10; E-7727/decitabine; Decitabine/E7727; ASTX-727 Approved Astex Pharmaceuticals Inc, National Cancer Institute INAQOVI, Inaqovi, Inqovi United States Myelodysplastic Syndromes Otsuka Pharmaceutical Co Ltd 2020-07-07 Leukemia, Myelogenous, Chronic; Leukemia; Solid tumours; Myelodysplastic Syndromes; Leukemia, Myelomonocytic, Chronic; Triple Negative Breast Neoplasms; Neoplasms; Mesothelioma; Pancytopenia; Leukemia, Myeloid, Acute; Glioma; Cytopenia; Metastatic breast cancer; Nervous System Neoplasms Details
Mecobalamin E-0302 Approved Methycobal, Naso B12, Myelogen, 悦敏兴, 弥尔神, 弥可保, 曲力, 奇信, ROZEALAMIN, NASOCOBAL, RHINOCOBAL Peripheral Nervous System Diseases; Autistic Disorder; Neuritis; Neuralgia; Vitamin B 12 Deficiency; Amyotrophic Lateral Sclerosis; Fibromyalgia Details
Azacitidine NSC-102816; 5-aza-CR; CC-486; NS-17; U-18496; NEX-18; NEX-18a Approved Celgene Corp 维达莎, Vidaza, Onureg United States Myelodysplastic Syndromes Bristol-Myers Squibb Company 2004-05-19 Leukemia, Myelomonocytic, Juvenile; Contracture; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Breast Neoplasms; Prostatic Neoplasms; Tuberculosis, Pulmonary; Brain Neoplasms; Sarcoma; Osteosarcoma; Hepatic Insufficiency; Primary Myelofibrosis; Leukemia, Myeloid, Acute; Multiple Myeloma; Thyroid Neoplasms; Lymphoma, Non-Hodgkin; Metastatic breast cancer; Lung Neoplasms; Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell; Carcinoma, Non-Small-Cell Lung; Leukemia, Large Granular Lymphocytic; Melanoma; Myelodysplastic-Myeloproliferative Diseases; Cerebral Palsy; Nasopharyngeal Neoplasms; Intestinal Neoplasms; Ependymoma; Leukemia, Myeloid; Lymphoma, T-Cell, Peripheral; Head and Neck Neoplasms; Solid tumours; Leukemia, Myelogenous, Chronic; Hematologic Neoplasms; Skin Melanoma; Carcinoma, Renal Cell; Squamous Cell Carcinoma of Head and Neck; Leukemia; Myelodysplastic Syndromes; Leukemia, Myelomonocytic, Chronic; Plasmacytoma; Neoplasms; Lymphoma, Large B-Cell, Diffuse; beta-Thalassemia; Hodgkin Disease; Glioblast Details
Triclabendazole EGA-230B; CGA-89317; NVP-EGA230 Approved Novartis Pharma Ag Egaten, Fasinex, Triclathera Iran Fascioliasis Novartis Pharma Ag 1989-01-01 Fascioliasis Details
Decitabine 5-aza-CdR; NSC-127716; AzadC; E-7373; DAC Approved Eisai Co Ltd Dacogen, 达珂 Mainland China Myelodysplastic Syndromes Mgi Pharma Inc 2006-05-02 Burkitt Lymphoma; Multiple Myeloma; Cycloplegia; Lymphoma, Mantle-Cell; Breast Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Lymphoma, Follicular; Neuroblastoma; Vulvar Neoplasms; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Colorectal Neoplasms; Primary Myelofibrosis; Leukemia, Myeloid, Acute; Thyroid Neoplasms; Adenocarcinoma, Follicular; Lymphoma; Lymphoma, Non-Hodgkin; Lung Neoplasms; Anemia, Sickle Cell; Myelodysplastic-Myeloproliferative Diseases; Precancerous Conditions; Carcinoma, Non-Small-Cell Lung; Breast Neoplasms, Male; Leukemia, Lymphocytic, Chronic, B-Cell; Neoplasm Metastasis; Melanoma; Thyroid Cancer, Papillary; Esophageal Neoplasms; Hematologic Neoplasms; Leukemia, Promyelocytic, Acute; Leukemia, Myeloid, Accelerated Phase; Leukemia; Lymphoma, B-Cell, Marginal Zone; Solid tumours; Purpura, Thrombocytopenic, Idiopathic; Liver Neoplasms; Erectile Dysfunction; Hypotension; Anaphylaxis; Thalassemia; Leukemia, Myelogenous, Chronic; Neutropenia; Myelodysplastic Syndromes; L Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Curcumin VOLT-03; VOLT-3; NSC-32982 Phase 3 Clinical University Of Pennsylvania Neuralgia; Lung Neoplasms; Lymphoma, T-Cell, Cutaneous; Adenocarcinoma, Mucinous; Cigarette Smoking; Cervical Intraepithelial Neoplasia; Cognitive Dysfunction; Uterine Cervical Dysplasia; Asthma; Osteoarthritis; Primary Myelofibrosis; Colorectal Neoplasms; Dentist-Patient Relations; Periapical Diseases; Prostatic Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tobacco Use Disorder; Oral Submucous Fibrosis; Thrombocythemia, Essential; Cognition Disorders; Uterine Cervical Neoplasms; Stomatitis; Neoplasm Metastasis; Macular Degeneration; Condylomata Acuminata; Carcinoma, Non-Small-Cell Lung; Aortic Aneurysm, Abdominal; Pancytopenia; Adenocarcinoma; Crohn Disease; Diabetes Mellitus; Hypogonadism; Renal Insufficiency, Chronic; Periodontitis; Lichen Planus, Oral; Diabetes Mellitus, Type 2; Neoplasms; Stomach Neoplasms; Spasm; Digestive System Diseases; Pain; Radiodermatitis; Gastritis, Atrophic; Depression; Myelodysplastic Syndromes; Metabolic Dysfunction-Associated Steatotic Liver Disease; Polycythemia Details
Azacitidine/Cedazuridine ASTX-030 Phase 3 Clinical Otsuka Pharmaceutical Co Ltd Leukemia, Myelogenous, Chronic; Myelodysplastic Syndromes; Leukemia, Myeloid, Acute Details
Guadecitabine Sodium SGI-110; S-110; 0RB89YH367 (UNII code) Phase 3 Clinical Otsuka Holdings Co Ltd Klatskin Tumor; Carcinoma, Hepatocellular; Adenocarcinoma; Paraganglioma; Carcinoma, Non-Small-Cell Lung; Melanoma; Gallbladder Neoplasms; Lung Neoplasms; Leukemia, Myeloid, Acute; Fallopian Tube Neoplasms; Colorectal Neoplasms; Gastrointestinal Stromal Tumors; Peritoneal Neoplasms; Cholangiocarcinoma; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Pancreatic Neoplasms; Myeloproliferative Disorders; Small Cell Lung Carcinoma; Carcinoma, Ovarian Epithelial; Carcinoma, Transitional Cell; Myelodysplastic Syndromes; Leukemia, Myelomonocytic, Chronic; Stomach Neoplasms; Pheochromocytoma; Carcinoma, Renal Cell; Chondrosarcoma; Kidney Neoplasms Details
EF-009 EF-009 Phase 2 Clinical Everfront Biotech Co Ltd Pancreatic Neoplasms Details
NTX-301 NTX-303 Phase 2 Clinical Southern Research Institute, Pinotbio Inc Solid tumours; Ovarian Neoplasms; Myelodysplastic Syndromes; Leukemia, Myelomonocytic, Chronic; Neoplasms; Carcinoma, Transitional Cell; Leukemia, Myeloid, Acute; Glioma Details
FdCyd NSC-48006; Ro-5-1090 Phase 2 Clinical City Of Hope National Medical Center, National Cancer Institute Head and Neck Neoplasms; Esophageal Neoplasms; Neoplasms; Mesothelioma; Urinary Bladder Neoplasms; Breast Neoplasms; Lung Neoplasms; Carcinoma, Non-Small-Cell Lung Details
Azacitidine (Boryung Pharmaceutical) Phase 2 Clinical Boryung Pharmaceutical Co Ltd Neoplasms Details
Decitabine/Tetrahydrouridine (EpiDestiny/Novo Nordisk) EPI-01; EPI01; NN 7533 Phase 2 Clinical Epicdestiny Anemia, Sickle Cell Details
GSK4172239D GSK-4172239-D Phase 1 Clinical Glaxosmithkline Plc Hematologic Diseases; Anemia, Sickle Cell Details

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