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GIPR

Brief Information

Name:Glucose-Dependent Insulinotropic Polypeptide Receptor
Target Synonym:Gastric inhibitory polypeptide receptor,GIPR,Glucose-Dependent Insulinotropic Polypeptide Receptor,GIP-R,PGQTL2
Number of Launched Drugs:1
Number of Drugs in Clinical Trials:31
Lastest Research Phase:Approved

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Part of Bioactivity data

CHEK-ATP208-Cell-based assay
 GIPR FACS

Expression analysis of human GIPR on HEK293/Human GIPR Stable Cell Line by FACS.
Cell surface staining using Alexa 647-labeled anti-human GIPR antibody was performed on HEK293/Human GIPR Stable Cell Line with different expression levels: HEK293/Human GIPR Stable Cell Line (Low Expression); HEK293/Human GIPR Stable Cell Line (Medium Expression); HEK293/Human GIPR Stable Cell Line (High Expression).

CHEK-ATP207-Cell-based assay
 GIPR FACS

Expression analysis of human GIPR on HEK293/Human GIPR Stable Cell Line by FACS.
Cell surface staining using Alexa 647-labeled anti-human GIPR antibody was performed on HEK293/Human GIPR Stable Cell Line with different expression levels: HEK293/Human GIPR Stable Cell Line (Low Expression); HEK293/Human GIPR Stable Cell Line (Medium Expression); HEK293/Human GIPR Stable Cell Line (High Expression).

GIR-H82E3-MALS-HPLC
GIPR MALS images

The purity of Biotinylated Human GIPR Protein, His,Avitag (Cat. No. GIR-H82E3) is more than 85% and the molecular weight of this protein is around 20-30 kDa verified by SEC-MALS.

GIR-H52D3-ELISA
 GIPR ELISA

Immobilized Human GIPR Protein, His,Flag Tag (Cat. No. GIR-H52D3) at 10 μg/mL (100 μL/well) on Nickel Coated plates (Cat. No. SP-19) can bind Anti-GIPR Antibody with a linear range of 1-63 ng/mL (QC tested).

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Tirzepatide LY-3298176; GIP/GLP-1 RA Approved Eli Lilly And Company Mounjaro, Zepbound, 穆峰达 United States Diabetes Mellitus, Type 2 Eli Lilly And Company 2022-05-13 Metabolic Diseases; Nutritional and Metabolic Diseases; Kidney Failure, Chronic; Diabetes Mellitus; Overweight; Renal Insufficiency, Chronic; Obesity; Alcoholism; Glucose Metabolism Disorders; Hepatic Insufficiency; Cardiovascular Diseases; Breast Neoplasms; Prostatic Neoplasms; Substance-Related Disorders; Sleep Apnea Syndromes; Endocrine System Diseases; Obesity, Morbid; Hypoglycemia; Opioid-Related Disorders; Sleep Apnea, Obstructive; Weight Gain; Metabolic Dysfunction-Associated Steatotic Liver Disease; Renal Insufficiency; Heart Failure; Diabetes Mellitus, Type 2; Diabetes Mellitus, Type 1 Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Retatrutide LY-3437943 Phase 3 Clinical Eli Lilly And Company Diabetes Mellitus, Type 2; Atherosclerosis; Renal Insufficiency; Sleep Apnea, Obstructive; Hepatic Insufficiency; Osteoarthritis, Knee; Cardiovascular Diseases; Renal Insufficiency, Chronic; Obesity; Overweight Details
BGM-0504 BGM-0504 Phase 3 Clinical Brightgene Bio-Medical Technology Co Ltd Diabetes Mellitus, Type 2; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Overweight Details
HRS-9531 HRS-9531; HRS9531 Phase 3 Clinical Fujian Suncadia Medicine Co Ltd Heart Failure, Diastolic; Diabetes Mellitus, Type 2; Polycystic Ovary Syndrome; Body Weight; Obesity; Overweight; Diabetes Mellitus Details
HS-20094 HS-20094 Phase 3 Clinical Jiangsu Hansoh Pharmaceutical Group Co Ltd Diabetes Mellitus, Type 2; Obesity; Overweight Details
CT-868 CT-868; RG-6641 Phase 2 Clinical Carmot Therapeutics Inc Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Obesity; Overweight Details
Efocipegtrutide HM-15211 Phase 2 Clinical Hanmi Pharmaceutical Co Ltd Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity Details
NNC0480-0389 NNC0480-0389 Phase 2 Clinical Novo Nordisk A/S Diabetes Mellitus, Type 2; Obesity; Overweight Details
HDM-1005 HDM-1005; HDM1005 Phase 2 Clinical Hangzhou Zhongmei Huadong Pharmaceutical Co Ltd Metabolic Dysfunction-Associated Steatotic Liver Disease; Diabetes Mellitus, Type 2; Obesity; Overweight Details
PF-07976016 PF-07976016 Phase 2 Clinical Pfizer Inc Obesity Details
NNC0519-0130 NNC0519-0130 Phase 2 Clinical Novo Nordisk A/S Diabetes Mellitus, Type 2; Obesity; Renal Insufficiency, Chronic Details
MWN-101 MWN-101 Phase 2 Clinical Shanghai Minwei Biotechnology Co Ltd Diabetes Mellitus, Type 2; Sleep Apnea, Obstructive; Obesity; Overweight Details
RAY-1225 RAY1225; RAY-1225 Phase 2 Clinical Guangdong Raynovent Biotech Co Ltd Diabetes Mellitus, Type 2; Metabolic Dysfunction-Associated Steatotic Liver Disease; Acute Kidney Injury; Hepatic Insufficiency; Obesity; Overweight Details
VK-2735 VK-2735 Phase 2 Clinical Viking Therapeutics Inc Weight Loss; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity Details
THDBH-120 THDBH120; THDBH121 Phase 2 Clinical Wuxi Apptec(Shanghai) Co Ltd Diabetes Mellitus, Type 2; Obesity; Overweight; Diabetes Mellitus Details
CT-388 CT-388; RG-6640 Phase 2 Clinical Carmot Therapeutics Inc Diabetes Mellitus, Type 2; Obesity; Overweight; Diabetes Mellitus Details
Maridebart cafraglutide AMG-133; AMG133 Phase 2 Clinical Amgen Inc Diabetes Mellitus, Type 2; Body Weight; Obesity; Overweight Details
LY-3493269 LY-3493269 Phase 1 Clinical Eli Lilly And Company Diabetes Mellitus, Type 2 Details
SCO-094 SCO-094; tak-094 Phase 1 Clinical Takeda Diabetes Mellitus, Type 2 Details
NN9542 NN9542; NN-9542 Phase 1 Clinical Novo Nordisk A/S Obesity Details
Gastric inhibitory polypeptide receptor agonist long acting II therapeutic (Eli Lilly and Company) Phase 1 Clinical Eli Lilly And Company Obesity; Diabetes Mellitus Details
NNC0650-0013 NNC0650-0013; NN9650; NN-9650 Phase 1 Clinical Novo Nordisk A/S Details
ZX-2010 ZX2010; ZX-2010 Phase 1 Clinical Jiangsu Zhongxin Pharmaceutical Co Ltd Diabetes Mellitus, Type 2; Obesity; Overweight Details
MWN-105 MWN-105 Phase 1 Clinical Shanghai Minwei Biotechnology Co Ltd Diabetes Mellitus, Type 2; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Overweight; Hyperlipidemias Details
ZX-2021 ZX2021; ZX-2021 Phase 1 Clinical Jiangsu Zhongxin Pharmaceutical Co Ltd Diabetes Mellitus, Type 2; Obesity; Overweight Details
HZ-012 DR-10628; HZ-012 Phase 1 Clinical Hangzhou Heze Pharmaceutical Technology Co Ltd, Zhejiang Doer Biologics Corp Metabolic Dysfunction-Associated Steatotic Liver Disease; Diabetes Mellitus, Type 2; Obesity; Diabetes Mellitus; Overweight Details
DR-10627 HZ-010; DR-10627 Phase 1 Clinical Hangzhou Heze Pharmaceutical Technology Co Ltd, Zhejiang Doer Biologics Corp Diabetes Mellitus, Type 2; Metabolic Dysfunction-Associated Steatotic Liver Disease; Diabetes Mellitus Details
Macupatide LY-3532226 Phase 1 Clinical Eli Lilly And Company Diabetes Mellitus, Type 1; Obesity Details
LY-3537031 LY3537031; LY-3537031 Phase 1 Clinical Eli Lilly And Company Obesity; Diabetes Mellitus Details
LY-3537021 LY-3537021 Phase 1 Clinical Eli Lilly And Company Diabetes Mellitus, Type 2 Details
GMA-106 GMA106; GMA-106 Phase 1 Clinical Gmax Biopharm Llc Obesity; Overweight Details
GIP[3-30]NH2 GIP[3-30]NH2 Copenhagen University Hospital Gentofte, University Of Copenhagen Details

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