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BCHE

Brief Information

Name:Butyrylcholinesterase
Target Synonym:BCHED,CHE2,E1,Butyrylcholinesterase,BuChE,EC:3.1.1.8,EC 3.1.1,BCHE,Acylcholine acylhydrolase,Pseudocholinesterase,Cholinesterase,CHE1,Cholinesterase (Serum) 2,Butyrylcholine Esterase,Choline Esterase II,Cholinesterase 1,EC 3.1.1.8
Number of Launched Drugs:2
Number of Drugs in Clinical Trials:2
Lastest Research Phase:Approved

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Cat. No. Species Product Description Structure Purity Feature
BHE-H52H3 Human Human BCHE / Butyrylcholinesterase Protein, His Tag (active enzyme)
BHE-H52H3-structure
BHE-H52H3-sds
ACRO Quality

Synonym Name

Acylcholine acylhydrolase; BCHE; Butyrylcholine esterase; Butyrylcholinesterase; CHE1; CHE1cholinesterase; Choline esterase II; cholinesterase 1; E1; EC 3.1.1.8; Pseudocholinesterase

Background

BCHE (also known as Butyrylcholinesterase,  pseudocholinesterase, plasma cholinesterase, or BuChE) is a nonspecific cholinesterase enzyme that hydrolyzes many different choline esters. Both acetylcholinesterase and butyrylcholinesterase represent therapeutic targets for ameliorating the cholinergic deficit considered to be responsible for the declines in cognitive, behavioral and global functioning characteristic of Alzheimer's disease (AD).

Clinical and Translational Updates

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Rivastigmine Tartrate SDZ-212-713; SDZ 212713; SDZ-ENA-713; ONO-2540; ENA-713; ENA-713D Approved Novartis Pharma Ag Exelon TDS, Rivastach, Exelon MR, Prometax, Exelon, 艾斯能 EU Parkinson Disease; Dementia; Alzheimer Disease Novartis Europharm Ltd 1998-05-11 Substance-Related Disorders; Brain Injuries, Traumatic; Down Syndrome; Delirium; Neurobehavioral Manifestations; Alzheimer Disease; Dementia; Parkinson Disease; Cocaine-Related Disorders; Dementia, Vascular; Cognition Disorders; Anticholinergic Syndrome Details
Rivastigmine transdermal patch (Luye Pharma) LY-03013; LY-30410; RID-TDS Approved Acino International AG Kingsmin, Rivirec Mainland China Alzheimer Disease Luye Pharma Group Ltd Alzheimer Disease; Parkinson Disease Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Bisnorcymserine ANVS-301 Phase 1 Clinical Horizon Therapeutics PLC Alzheimer Disease Details

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